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Search Results for " bradykinin receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
TP1181 Bradykinin (2-9) Des-Arg1-bradykinin Bradykinin Receptor
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P.
TP1445 [Des-Arg9]-Bradykinin acetate Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.
TP1277 Bradykinin Endogenous Metabolite , Bradykinin Receptor
Bradykinin is an inflammatory mediator. It is a peptide that causes blood vessels to dilate (enlarge) via the release of prostacyclin, nitric oxide, and Endothelium-Derived Hyperpolarizing Factor. Bradykinin is a physiol...
T5048 SSR240612 Bradykinin Receptor
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors, respectively).
T22344 Icatibant Acetate Bradykinin Receptor
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.
T2086 ELN-441958 ELN 441958 Bradykinin Receptor
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958(ELN 441958) is highly selective for B1 over B2 receptors.
T7645 [Des-Arg9]-Bradykinin [Des-Arg9]-Bradykinin(2TFA) Bradykinin Receptor
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
TP2268L Lys-Bradykinin acetate(342-10-9 free base) Bradykinin Receptor
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
T8809 [Des-Arg9]-Bradykinin TFA Bradykinin Receptor
[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
T33421 MK-0686 MK0686 Bradykinin Receptor
MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.
T36442L (Hyp³)-Bradykinin acetate (Hyp³)-Bradykinin acetate (37642-65-2 Free base) Bradykinin Receptor
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.
TP2075L Bombinakinin M acetate Bombinakinin M acetate(509151-65-9 free base) Bradykinin Receptor
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is approximately 50 times more potent than bradykinin.
TP1918L1 Lys-[Des-Arg9]Bradykinin acetate Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces p...
TP1918L Lys-[Des-Arg9]Bradykinin,TFA Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa) Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripher...
T34485 Safotibant LF220542,LF 220542,LF 22-0542,LF-220542,LF-22-0542,LF22-0542 Bradykinin Receptor
Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema.
TP1917L1 Sar-[D-Phe8]-des-Arg9-Bradykinin acetate Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to aminopeptidase, kininase I and II (ACE) and neutral endopeptidase cl...
T26627L Anatibant 2HCl Anatibant 2HCl(209733-45-9 Free base) Bradykinin Receptor
Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
TP1933 R715 TFA(185052-09-9 free base) R 715 Bradykinin Receptor
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49). Displays no activity at B2 receptors. Reduces mechanical hypernociception in a mouse model of neuropathic pain. Me...
TP1931L1 [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base) cholecystokinin
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist ...
T4200 Sacubitril hemicalcium salt AHU-377 (hemicalcium salt),AHU377 calcium salt Neprilysin
Sacubitril hemicalcium salt (AHU377 calcium salt) is a potent NEP inhibitor with an IC50 of 5 nM. Sacubitril hemicalcium salt is a component of the heart failure medicine LCZ696. Sacubitril hemicalcium salt is a prodrug ...

Compounds

Bradykinin (2-9)
TP1181
Synonym: Des-Arg1-bradykinin
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin acetate
TP1445
Synonym:
Target: Bradykinin Receptor
Bradykinin
TP1277
Synonym:
Target: Endogenous Metabolite, Bradykinin Receptor
SSR240612
T5048
Synonym:
Target: Bradykinin Receptor
Icatibant Acetate
T22344
Synonym:
Target: Bradykinin Receptor
ELN-441958
T2086
Synonym: ELN 441958
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin
T7645
Synonym: [Des-Arg9]-Bradykinin(2TFA)
Target: Bradykinin Receptor
Lys-Bradykinin acetate(342-10-9 free base)
TP2268L
Synonym:
Target: Bradykinin Receptor
[Des-Arg9]-Bradykinin TFA
T8809
Synonym:
Target: Bradykinin Receptor
MK-0686
T33421
Synonym: MK0686
Target: Bradykinin Receptor
(Hyp³)-Bradykinin acetate
T36442L
Synonym: (Hyp³)-Bradykinin acetate (37642-65-2 Free base)
Target: Bradykinin Receptor
Bombinakinin M acetate
TP2075L
Synonym: Bombinakinin M acetate(509151-65-9 free base)
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin acetate
TP1918L1
Synonym: Lys-[Des-Arg9]Bradykinin acetate (71800-36-7 free base)
Target: Bradykinin Receptor
Lys-[Des-Arg9]Bradykinin,TFA
TP1918L
Synonym: Lys-[Des-Arg9]Bradykinin,TFA 71800-36-7(fb-tfa)
Target: Bradykinin Receptor
Safotibant
T34485
Synonym: LF220542,LF 220542,LF 22-0542,LF-220542,LF-22-0542,LF22-0542
Target: Bradykinin Receptor
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
TP1917L1
Synonym: Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base)
Target: Bradykinin Receptor
Anatibant 2HCl
T26627L
Synonym: Anatibant 2HCl(209733-45-9 Free base)
Target: Bradykinin Receptor
R715 TFA(185052-09-9 free base)
TP1933
Synonym: R 715
Target: Bradykinin Receptor
[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
TP1931L1
Synonym: [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate(96736-12-8 free base)
Target: cholecystokinin
Sacubitril hemicalcium salt
T4200
Synonym: AHU-377 (hemicalcium salt),AHU377 calcium salt
Target: Neprilysin
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TargetMol